DE69837684D1 - Verfahren zur selektiven Derivatisierung von Taxanen - Google Patents

Verfahren zur selektiven Derivatisierung von Taxanen

Info

Publication number
DE69837684D1
DE69837684D1 DE69837684T DE69837684T DE69837684D1 DE 69837684 D1 DE69837684 D1 DE 69837684D1 DE 69837684 T DE69837684 T DE 69837684T DE 69837684 T DE69837684 T DE 69837684T DE 69837684 D1 DE69837684 D1 DE 69837684D1
Authority
DE
Germany
Prior art keywords
sup
taxanes
hydroxytaxane
acyloxy
selective derivatization
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69837684T
Other languages
English (en)
Other versions
DE69837684T2 (de
Inventor
Robert A Holton
Paul A Clark
Zhuming Zhang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Florida State University
Original Assignee
Florida State University
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27368950&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE69837684(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Florida State University filed Critical Florida State University
Application granted granted Critical
Publication of DE69837684D1 publication Critical patent/DE69837684D1/de
Publication of DE69837684T2 publication Critical patent/DE69837684T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C07F7/1872—Preparation; Treatments not provided for in C07F7/20
    • C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888
DE69837684T 1997-08-18 1998-08-17 Verfahren zur selektiven Derivatisierung von Taxanen Expired - Lifetime DE69837684T2 (de)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US5600097P 1997-08-18 1997-08-18
US56000 1997-08-18
US8126598P 1998-04-09 1998-04-09
US81265 1998-04-09
US63477 1998-04-20
US09/063,477 US7288665B1 (en) 1997-08-18 1998-04-20 Process for selective derivatization of taxanes

Publications (2)

Publication Number Publication Date
DE69837684D1 true DE69837684D1 (de) 2007-06-06
DE69837684T2 DE69837684T2 (de) 2007-09-06

Family

ID=27368950

Family Applications (3)

Application Number Title Priority Date Filing Date
DE69836072T Expired - Lifetime DE69836072T2 (de) 1997-08-18 1998-08-17 Verfahren zur selektiven derivatisierung von taxanen
DE69837684T Expired - Lifetime DE69837684T2 (de) 1997-08-18 1998-08-17 Verfahren zur selektiven Derivatisierung von Taxanen
DE69834584T Expired - Fee Related DE69834584T2 (de) 1997-08-18 1998-08-17 Verfahren zur selektiven Derivatisierung von Taxanen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE69836072T Expired - Lifetime DE69836072T2 (de) 1997-08-18 1998-08-17 Verfahren zur selektiven derivatisierung von taxanen

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE69834584T Expired - Fee Related DE69834584T2 (de) 1997-08-18 1998-08-17 Verfahren zur selektiven Derivatisierung von Taxanen

Country Status (25)

Country Link
US (5) US7288665B1 (de)
EP (6) EP1795528A1 (de)
JP (1) JP2001504864A (de)
KR (1) KR100596989B1 (de)
CN (3) CN1205196C (de)
AT (3) ATE326455T1 (de)
AU (1) AU744987B2 (de)
BR (1) BR9806145A (de)
CA (2) CA2597799A1 (de)
CY (1) CY1105399T1 (de)
CZ (1) CZ296580B6 (de)
DE (3) DE69836072T2 (de)
DK (3) DK0956284T3 (de)
ES (3) ES2259646T3 (de)
HU (1) HUP0300425A3 (de)
ID (1) ID21654A (de)
IL (3) IL129386A0 (de)
NO (4) NO325139B1 (de)
NZ (1) NZ335156A (de)
PL (3) PL201641B1 (de)
PT (3) PT1170292E (de)
RU (1) RU2225402C2 (de)
SG (1) SG97986A1 (de)
WO (1) WO1999009021A1 (de)
ZA (1) ZA987394B (de)

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NO325139B1 (no) 2008-02-11
DE69837684T2 (de) 2007-09-06
EP1170292A3 (de) 2002-04-03
DE69834584D1 (de) 2006-06-22
JP2001504864A (ja) 2001-04-10
KR100596989B1 (ko) 2006-07-07
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US20050272944A1 (en) 2005-12-08
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BR9806145A (pt) 2000-01-18
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AU9021198A (en) 1999-03-08
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